Thomas Blacklock : rechercher sur Z-Library

Organic Process Research & Development

Année:

2001

Langue:

english

Fichier:

PDF, 188 KB

english, 2001

CO 2 Offgas as a Mechanistic Probe and Scale-up Tool in N-Acylations Using Mixed Anhydrides from Amino Acids and Isobutyl Chloroformate

Chaudhary, Apurva, Girgis, Michael J., Prashad, Mahavir, Hu, Bin, Har, Denis, Repič, Oljan, Blacklock, Thomas J.

Journal:

Année:

2003

Langue:

english

Fichier:

PDF, 132 KB

english, 2003

A Practical and Chemoselective Reduction of Nitroarenes to Anilines Using Activated Iron

Yugang Liu, Yansong Lu, Mahavir Prashad, Oljan Repič, Thomas J. Blacklock

Journal:

Année:

2005

Langue:

english

Fichier:

PDF, 64 KB

english, 2005

Dual Nucleophilic Catalysis with DABCO for the N-Methylation of Indoles.

Wen-Chung Shieh, Steven Dell, Andrew Bach, Oljan Repic, Thomas J. Blacklock

Journal:

Année:

2003

Fichier:

PDF, 136 KB

2003

Selective deprotection of alkyl t-butyldimethylsilyl ethers in the presence of aryl t-butyldimethylsilyl ethers with bismuth bromide

Joginder S. Bajwa, James Vivelo, Joel Slade, Oljan Repič, Thomas Blacklock

Journal:

Liu, Yugang, Shen, Lichun, Prashad, Mahavir, Tibbatts, Jessica, Repič, Oljan, Blacklock, Thomas J.

Année:

2000

Langue:

english

Fichier:

PDF, 173 KB

english, 2000

An efficient large scale resolution of (±)-threo-methylphenidate hydrochloride (Ritalin® hydrochloride)

Mahavir Prashad, Denis Har, Oljan Repic, Thomas J. Blacklock, Peter Giannousis

Journal:

Tetrahedron: Asymmetry

Année:

1999

Langue:

english

Fichier:

PDF, 150 KB

english, 1999

A Green N-Detosylation of Indoles and Related Heterocycles Using Phase Transfer Catalysis

Journal:

Organic Process Research & Development

Année:

2008

Langue:

english

Fichier:

PDF, 89 KB

english, 2008

LCZ696: a dual-acting sodium supramolecular complex

Lili Feng, Piotr H. Karpinski, Paul Sutton, Yugang Liu, David F. Hook, Bin Hu, Thomas J. Blacklock, Philip E. Fanwick, Mahavir Prashad, Sven Godtfredsen, Christoph Ziltener

Journal:

Shieh, Wen-Chung, Dell, Steven, Bach, Andrew, Repič, Oljan, Blacklock, Thomas J.

Année:

2012

Langue:

english

Fichier:

PDF, 254 KB

english, 2012

Dual Nucleophilic Catalysis with DABCO for the N-Methylation of Indoles

Journal:

Journal of Organic Chemistry

Année:

2003

Langue:

english

Fichier:

PDF, 77 KB

english, 2003

Synthesis of semisynthetic dipeptides using N-carboxyanhydrides and chiral induction on Raney nickel. A method practical for large scale

Blacklock, Thomas J., Shuman, Richard F., Butcher, John W., Shearin, Willard E., Budavari, John, Grenda, Victor J.

Journal:

Journal of Organic Chemistry

Année:

1988

Langue:

english

Fichier:

PDF, 1.09 MB

english, 1988

Process Development of a Large-Scale Synthesis of TKA731: A Tachykinin Receptor Antagonist

Prashad, Mahavir, Har, Denis, Hu, Bin, Kim, Hong-Yong, Girgis, Michael J., Chaudhary, Apurva, Repič, Oljan, Blacklock, Thomas J., Marterer, Wolfgang

Journal:

Organic Process Research & Development

Année:

2004

Langue:

english

Fichier:

PDF, 171 KB

english, 2004

A New Reaction of Aminoiminomethanesulfonic Acid with Methyl Anthranilates

Prashad, Mahavir, Chen, Lijian, Repic, Oljan, Blacklock, Thomas J.

Journal:

Synthetic Communications

Année:

1998

Langue:

english

Fichier:

PDF, 162 KB

english, 1998

Quantifying and Reducing International Space Station Vulnerability Following Orbital Debris Penetration

Williamsen, Joel, Blacklock, Kevin, Evans, Hilary J., Guay, Thomas D.

Journal:

Journal of Spacecraft and Rockets

Année:

1999

Langue:

english

Fichier:

PDF, 827 KB

english, 1999

New Trends in Palladium-Catalyzed Transfer Hydrogenations Using Formic Acid

Kapa Prasad, Xinglong Jiang, Joel S. Slade, Jennifer Clemens, Oljan Repič, Thomas J. Blacklock

Journal:

George T. Lee, Xinglong Jiang, Kapa Prasad, Oljan Repič, Thomas J. Blacklock

Année:

2005

Langue:

english

Fichier:

PDF, 81 KB

english, 2005

Pd-Catalyzed ortho-Selective Oxidative Coupling of Halogenated Acetanilides with Acrylates

Journal:

Année:

2005

Langue:

english

Fichier:

PDF, 86 KB

english, 2005

ChemInform Abstract: A Convenient and Practical Method for N-Acylation of 2-Oxazolidinone Chiral Auxiliaries with Acids.

Mahavir Prashad, Hong-Yong Kim, Denis Har, Oljan Repic, Thomas J. Blacklock

Journal:

Année:

1999

Fichier:

PDF, 28 KB

1999

ChemInform Abstract: An Improved and Practical Sharpless Oxidation of Primary Alcohols to the Carboxylic Acids.

Mahavir Prashad, Yansong Lu, Hong-Yong Kim, Bin Hu, Iljan Repic, Thomas J. Blacklock

Journal:

Année:

1999

Fichier:

PDF, 31 KB

1999

ChemInform Abstract: Mild and Regioselective Oxidative Bromination of Anilines Using Potassium Bromide and Sodium Perborate.

Didier Roche, Kapa Prasad, Oljan Repic, Thomas J. Blacklock

Journal:

Année:

2000

Fichier:

PDF, 28 KB

2000

ChemInform Abstract: β-Hydrogen-Containing Sodium Alkoxides as Suitable Bases in Palladium-Catalyzed Aminations of Aryl Halides.

Mahavir Prashad, Bin Hu, Yansong Lu, Robert Draper, Denis Har, Oljan Repic, Thomas J. Blacklock

Journal:

Année:

2000

Fichier:

PDF, 35 KB

2000

ChemInform Abstract: Selective Deprotection of Alkyl t-Butyldimethylsilyl Ethers in the Presence of Aryl t-Butyldimethylsilyl Ethers with Bismuth Bromide.

Joginder S. Bajwa, James Vivelo, Joel Slade, Oljan Repic, Thomas Blacklock

Journal:

Année:

2000

Fichier:

PDF, 29 KB

2000

ChemInform Abstract: A New, Convenient and Selective 4-Dimethylaminopyridine-Catalyzed Trifluoroacetylation of Anilines with Ethyl Trifluoroacetate.

Mahavir Prashad, Bin Hu, Denis Har, Oljan Repic, Thomas J. Blacklock

Journal:

Année:

2001

Fichier:

PDF, 32 KB

2001

ChemInform Abstract: A Mild Method for Ring-Opening Aminolysis of Lactones.

Wenming Liu, David D. Xu, Oljan Repic, Thomas J. Blacklock

Journal:

Wenming Liu, Joanna M. Szewczyk, Liladhar Waykole, Oljan Repic, Thomas J. Blacklock

Année:

2001

Fichier:

PDF, 30 KB

2001

ChemInform Abstract: Total Synthesis of Bengamide E.

Journal:

Wen-Chung Shieh, Ratna Shekhar, Thomas Blacklock, Anthony Tedesco

Année:

2002

Fichier:

PDF, 31 KB

2002

ChemInform Abstract: A Simple, Recyclable, Polymer-Supported Palladium Catalyst for Suzuki Coupling — An Effective Way to Minimize Palladium Contamination.

Journal:

Année:

2002

Fichier:

PDF, 29 KB

2002

In situ Generation of Et3SiBr from BiBr3 and Et3SiH and Its Use in Preparation of Dialkyl Ethers.

Joginder S. Bajwa, Xinglong Jiang, Joel Slade, Kapa Prasad, Oljan Repic, Thomas J. Blacklock

Journal:

Année:

2002

Fichier:

PDF, 34 KB

2002

Double Heck Reaction of Bridged o,o′-Dibromobiaryls with Ethyl Acrylate.

Mahavir Prashad, Yugang Liu, Xiao Yin Mak, Denis Har, Oljan Repic, Thomas J. Blacklock

Journal:

Année:

2003

Fichier:

PDF, 124 KB

2003

An Efficient and Large-Scale Enantioselective Synthesis of PNP405 (I): A Purine Nucleoside Phosphorylase Inhibitor.

Mahavir Prashad, Denis Har, Lijian Chen, Hong-Yong Kim, Oljan Repic, Thomas J. Blacklock

Journal:

Année:

2003

Fichier:

PDF, 60 KB

2003

Etherification of Alkoxydialkylsilanes with Carbonyl Compounds.

Xinglong Jiang, Joginder S. Bajwa, Joel Slade, Kapa Prasad, Oljan Repic, Thomas J. Blacklock

Journal:

Année:

2003

Fichier:

PDF, 120 KB

2003

An Efficient and Practical N-Methylation of Amino Acid Derivatives.

Mahavir Prashad, Denis Har, Bin Hu, Hong-Yong Kim, Oljan Repic, Thomas J. Blacklock

Journal:

Wenming Liu, Joanna Szewczyk, Liladhar Waykole, Oljan Repic, Thomas J. Blacklock

Année:

2003

Fichier:

PDF, 21 KB

2003

Practical Synthesis of Diaryloxymethanes.

Journal:

Année:

2003

Fichier:

PDF, 72 KB

2003

DABCO- and DBU-Accelerated Green Chemistry for N-, O-, and S-Benzylation with Dibenzyl Carbonate.

Wen-Chung Shieh, Mario Lozanov, Mauricio Loo, Oljan Repic, Thomas J. Blacklock

Journal:

Wenming Liu, Joanna Szewczyk, Liladhar Waykole, Oljan Repic, Thomas J. Blacklock

Année:

2003

Fichier:

PDF, 122 KB

2003

Practical Synthesis of Diaryloxymethanes.

Journal:

Yugang Liu, Mahavir Prashad, Oljan Repic, Thomas J. Blacklock

Année:

2003

Fichier:

PDF, 71 KB

2003

Palladium-Catalyzed Amination with Benzophenone Imine as a New, Safe and Practical Alternative to Nitration for the Synthesis of 7-Amino-2,1,3-benzothiadiazoles.

Journal:

Lech Ciszewski, Daquiang Xu, Oljan Repic, Thomas J. Blacklock

Année:

2004

Fichier:

PDF, 105 KB

2004

Reductive Alkylation of Thioureas: A Highly Practical Synthesis of Unsymmetrical N,N′-Disubstituted Thioureas.

Journal:

Année:

2005

Fichier:

PDF, 20 KB

2005

A General and Facile Synthesis of 1,3-Diaryl-4-pyrazoleacetic Acid Esters.

David D. Xu, George T. Lee, Xinglong Jiang, Kapa Prasad, Oljan Repic, Thomas J. Blacklock

Journal:

Année:

2005

Fichier:

PDF, 20 KB

2005

1,2,3-Triazole as a Safer and Practical Substitute for Cyanide in the Bruylants Reaction for the Synthesis of Tertiary Amines Containing Tertiary Alkyl or Aryl Groups.

Mahavir Prashad, Yugang Liu, Denis Har, Oljan Repic, Thomas J. Blacklock

Journal:

Yugang Liu, Mahavir Prashad, Oljan Repič, Thomas J. Blacklock

Année:

2005

Fichier:

PDF, 23 KB

2005

Palladium-catalyzed amination with benzophenone imine as a new, safe and practical alternative to nitration for the synthesis of 7-amino-2,1,3-benzothiadiazoles

Journal:

Année:

2003

Langue:

english

Fichier:

PDF, 31 KB

english, 2003

A general and facile synthesis of 1,3-diaryl-4-pyrazoleacetic acid esters

David D. Xu, George T. Lee, Xinglong Jiang, Kapa Prasad, Oljan Repic, Thomas J. Blacklock

Journal:

Année:

2005

Langue:

english

Fichier:

PDF, 84 KB

english, 2005

Lithiation of N-protected-dihydro-1,4-benzoxaziness

Yansong J. Lu, Bin Hu, Mahavir Prashad, Shaum Kabadi, Oljan Repič, Thomas J. Blacklock

Journal:

Année:

2006

Langue:

english

Fichier:

PDF, 77 KB

english, 2006

A general synthesis of 8-hydroxy-6-substituted-1,7-naphthyridines

Xinglong Jiang, Guang-Pei Chen, Kapa Prasad, Oljan Repič, Thomas J. Blacklock

Journal:

Année:

2006

Langue:

english

Fichier:

PDF, 220 KB

english, 2006

Ethyl trifluoroacetate: a powerful reagent for differentiating amino groups

Daqiang Xu, Kapa Prasad, Oljan Repic, Thomas J. Blacklock

Journal:

Année:

1995

Langue:

english

Fichier:

PDF, 229 KB

english, 1995

An expeditious synthesis of a biscyclam with an aromatic linker

Daqiang Xu, Paul G. Mattner, Kapa Prasad, Oljan Repic, Thomas J. Blacklock

Journal:

Orin Tempkin, Thomas J. Blacklock, J. Andrew Burke, Maria Anastasia

Année:

1996

Langue:

english

Fichier:

PDF, 191 KB

english, 1996

β-butyrolactone as a chiral building block in organic synthesis: A convenient synthesis of MK-0507 keto sulfone

Journal:

Tetrahedron: Asymmetry

Année:

1996

Langue:

english

Fichier:

PDF, 249 KB

english, 1996

Reductive alkylation of thioureas: a highly practical synthesis of unsymmetrical N,N′-disubstituted thioureas

Lech Ciszewski, Daquiang Xu, Oljan Repič, Thomas J. Blacklock

Journal:

Année:

2004

Langue:

english

Fichier:

PDF, 245 KB

english, 2004

1,2,3-Triazole as a safer and practical substitute for cyanide in the Bruylants reaction for the synthesis of tertiary amines containing tertiary alkyl or aryl groups

Mahavir Prashad, Yugang Liu, Denis Har, Oljan Repič, Thomas J. Blacklock

Journal:

Année:

2005

Langue:

english

Fichier:

PDF, 95 KB

english, 2005

Deprotection of heteroaromatic carbamates via a base-catalyzed methanolysis

Wen-Chung Shieh, Song Xue, Joe McKenna, Kapa Prasad, Oljan Repič, Thomas Blacklock

Journal:

Joginder S. Bajwa, Guang-Pei Chen, Kapa Prasad, Oljan Repič, Thomas J. Blacklock

Année:

2006

Langue:

english

Fichier:

PDF, 98 KB

english, 2006

Deprotection of N-tosylated indoles and related structures using cesium carbonate

Journal:

Année:

2006

Langue:

english

Fichier:

PDF, 92 KB

english, 2006

A new reaction of N-aryl-2-pyrimidinamines with triphosgene

Mahavir Prashad, Bin Hu, Hong-Yong Kim, Denis Har, Oljan Repič, Thomas J. Blacklock

Journal:

Année:

2007

Langue:

english

Fichier:

PDF, 110 KB

english, 2007

Mild and regioselective oxidative bromination of anilines using potassium bromide and sodium perborate

Didier Roche, Kapa Prasad, Oljan Repic, Thomas J Blacklock

Journal:

Année:

2000

Langue:

english

Fichier:

PDF, 110 KB

english, 2000

A new, convenient and selective 4-dimethylaminopyridine-catalyzed trifluoroacetylation of anilines with ethyl trifluoroacetate

Mahavir Prashad, Bin Hu, Denis Har, Oljan Repič, Thomas J Blacklock

Journal: